平安! 发表于 2011-11-9 19:57
& b( j% C# ^+ Y+ k* i4 B$ \3 oPazopanib (100 mg/kg/day free base equivalent) 4 l% _( p7 ^1 @% b- b) R9 y, Q8 v& n1 U( i
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。" y: G$ [5 C$ ]2 a1 k2 d& X7 b
搜索了一下,原料一大堆。0 L- H8 B1 w7 ^( I. L
7 u7 x" P# v9 ^# b对不起!100mg/kg是用于移植瘤的,我弄错了。6 e& l7 W% H# n0 p/ V
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以下是正版说明书的推荐用量。" F& Q1 D6 p. F. ^
; ?* r6 X9 p+ P2 a* s--------------------- DOSAGE AND ADMINISTRATION ----------------* J& G. P" O1 r+ J6 b1 S
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
_! R1 x$ q. Q5 T4 s* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
6 O; H( h( I, t. F4 m q8 c) u% k---------------------DOSAGE FORMS AND STRENGTHS --------------
7 T/ W( P. T) _200 mg tablets. (3) y- o0 ^" Q* Q+ W0 x& p# M y
-------------------------------CONTRAINDICATIONS------------------------ |