平安! 发表于 2011-11-9 19:57
; C) V5 Z2 h! E6 F6 MPazopanib (100 mg/kg/day free base equivalent)
; [9 g" |0 N1 T0 o 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
' \2 f" z; J& f3 z- c搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。2 |% {0 E, D0 z. c! C3 _* `, g
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以下是正版说明书的推荐用量。8 V, _4 w8 b% e) b* y) \
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--------------------- DOSAGE AND ADMINISTRATION ----------------1 F. u) e5 n; S
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) 6 l5 ?- \0 W0 K% C ~
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) / N3 v) y' X* a7 o' {
---------------------DOSAGE FORMS AND STRENGTHS --------------6 ^1 `/ L4 Y! ^ ^4 V* K# x/ s6 U
200 mg tablets. (3) 4 p* B, n, q3 m+ p3 M
-------------------------------CONTRAINDICATIONS------------------------ |